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Early Drug-Discovery Efforts towards the Identification of EP300/CBP Histone Acetyltransferase (HAT) Inhibitors
Authors:Dr Annissa J Huhn  Dr Anna S Gardberg  Florence Poy  Dr Francois Brucelle  Dr Valerie Vivat  Nico Cantone  Gaurav Patel  Dr Chirag Patel  Dr Richard Cummings  Dr Robert Sims  Dr Julian Levell  Dr James E Audia  Dr Archana Bommi-Reddy  Dr Jonathan E Wilson
Affiliation:1. Constellation Pharmaceuticals, 215 First Street, Cambridge, MA 02142;2. Foghorn Therapeutics, 100 Binney St., Cambridge, MA 02142;3. Piramal Enterprises Limited-Discovery Solutions Ahmedabad, Gujarat, 382 213;4. Third Rock Ventures, 29 Newbury St. #301, Boston, MA 02116
Abstract:
Keywords:CBP  EP300  epigenetics  histone acetyltransferase
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