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Synthesis and Biological Evaluation of New Triazolo‐ and Imidazolopyridine RORγt Inverse Agonists
Authors:Dr. Samuel Hintermann  Dr. Christine Guntermann  Dr. Henri Mattes  Dr. David A. Carcache  Dr. Juergen Wagner  Dr. Anna Vulpetti  Dr. Andreas Billich  Dr. Janet Dawson  Dr. Klemens Kaupmann  Dr. Joerg Kallen  Dr. Rowan Stringer  Dr. David Orain
Affiliation:1. Global Discovery Chemistry, Novartis Institutes for BioMedical Research, Basel, Switzerland;2. ATI, Novartis Institutes for BioMedical Research, Basel, Switzerland;3. CPC, Novartis Institutes for BioMedical Research, Basel, Switzerland;4. MAP, Novartis Institutes for BioMedical Research, Basel, Switzerland
Abstract:
Keywords:imidazopyridines  inverse agonists  oxadiazoles  plasma protein binding  RORγ  t
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