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Sylvain Petit Yann Duroc Dr. Valéry Larue Dr. Carmela Giglione Dr. Carole Léon Dr. Coralie Soulama Dr. Alexis Denis Dr. Frédéric Dardel Prof. Thierry Meinnel Dr. Isabelle Artaud Dr. 《ChemMedChem》2009,4(2):133-133
The cover picture shows a “reverse” indole derivative in complex with Bacillus stearothermophilus peptide deformylase (PDF). This compound was selected from a structure–activity relationship study as a potent inhibitor of bacterial PDFs and shows antibacterial activity toward Bacillus subtilis as well as other pathogens such as Streptococcus pneumoniae and Staphylococcus aureus. For more details, see the Full Paper by I. Artaud et al. on p. 261 ff.
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Dr. Stefan Peukert Dr. Feng He Miao Dai Rui Zhang Yingchuan Sun Dr. Karen Miller‐Moslin Michael McEwan Dr. Bharat Lagu Kate Wang Dr. Naeem Yusuff Aaron Bourret Arun Ramamurthy Dr. Wieslawa Maniara Adam Amaral Anthony Vattay Anlai Wang Ribo Guo Jing Yuan John Green Dr. Juliet Williams Dr. Silvia Buonamici Dr. Joseph F. Kelleher III Dr. Marion Dorsch 《ChemMedChem》2013,8(8):1229-1229
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Hartmut Schirok Dr. Raimund Kast Dr. Santiago Figueroa‐Pérez Dr. Samir Bennabi Dr. Mark J. Gnoth Dr. Achim Feurer Dr. Heike Heckroth Dr. Michael Thutewohl Dr. Holger Paulsen Dr. Andreas Knorr Dr. Joachim Hütter Dr. Mario Lobell Dr. Klaus Münter Dr. Volker Geiß Dr. Heimo Ehmke Prof. Dr. Dieter Lang Dr. Martin Radtke Dr. Joachim Mittendorf Dr. Johannes‐Peter Stasch Dr. 《ChemMedChem》2008,3(12):1797-1797
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Cover Picture: Covalent Inhibition of HIV‐1 Integrase by N‐Succinimidyl Peptides (ChemMedChem 18/2016) 下载免费PDF全文
Dr. Koushik Chandra Dr. Priyadip Das Dr. Samarasimhareddy Mamidi Dr. Mattan Hurevich Anat Iosub‐Amir Dr. Norman Metanis Dr. Meital Reches Prof. Assaf Friedler 《ChemMedChem》2016,11(18):1969-1969
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Cover Picture: Detection of Human α‐L‐Fucosidases by a Quinone Methide‐Generating Probe: Enhanced Activities in Response to Helicobacter pylori Infection (ChemBioChem 11/2015) 下载免费PDF全文
Manjula Nandakumar Yu‐Ling Hsu Jason C.‐Y Lin Chun Lo Prof. Lee‐Chiang Lo Prof. Chun‐Hung Lin 《Chembiochem : a European journal of chemical biology》2015,16(11):1525-1525
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Sylvain Petit Yann Duroc Dr. Valéry Larue Dr. Carmela Giglione Dr. Carole Léon Dr. Coralie Soulama Dr. Alexis Denis Dr. Frédéric Dardel Prof. Thierry Meinnel Dr. Isabelle Artaud Dr. 《ChemMedChem》2009,4(2):261-275
SAR by NMR : A series of indole compounds derived from 5‐bromo‐1H‐indole‐3‐acetohydroxamic acid were synthesized. Their inhibitory activities were evaluated against purified peptide deformylases (PDFs), and their antibacterial activities against B. subtilis, E. coli (wild type and tolC), and a variety of pathogens were also determined. The potency of the best inhibitors was related to the NMR footprints of the respective acids with 15N‐labeled E. coli Ni‐PDF.
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