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Screening of Various Hormone‐Sensitive Lipase Inhibitors as Endocannabinoid‐Hydrolyzing Enzyme Inhibitors
Authors:Anna Minkkilä  Juha R Savinainen Dr  Heikki Käsnänen  Henri Xhaard Dr  Tapio Nevalainen Dr  Jarmo T Laitinen Dr  Antti Poso Prof Dr  Jukka Leppänen Dr  Susanna M Saario Dr
Affiliation:1. Department of Pharmaceutical Chemistry, University of Kuopio, P.O.Box 1627, 70211 Kuopio (Finland), Fax: (+358)?17‐162‐252;2. Institute of Biomedicine/Physiology, University of Kuopio, P.O.Box 1627, FI‐70211 Kuopio (Finland);3. Division of Pharmaceutical Chemistry and Centre for Drug Research, University of Helsinki, P.O.Box 56, 00014 Helsinki (Finland);4. The Skaggs Institute for Chemical Biology and Department of Chemical Physiology, The Scripps Research Institute, 10550 North Torrey Pines Road, La Jolla, California 92037 (USA)
Abstract:
Keywords:drug discovery  drug design  molecular modeling  inhibitors  enzymes  FAAH  HSL  MGL
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