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Front Cover: Deciphering Specificity Determinants for FR900359‐Derived Gqα Inhibitors Based on Computational and Structure–Activity Studies (ChemMedChem 16/2018)
Authors:Raphael Reher  Dr Toni Kühl  Suvi Annala  Tobias Benkel  Desireé Kaufmann  Britta Nubbemeyer  Justin Patrick Odhiambo  Dr Pascal Heimer  Charlotte Anneke Bäuml  Dr Stefan Kehraus  Dr Max Crüsemann  Prof Dr Evi Kostenis  Dr Daniel Tietze  Prof Dr Gabriele M König  Prof Dr Diana Imhof
Affiliation:1. Institute of Pharmaceutical Biology, University of Bonn, Bonn, Germany;2. Pharmaceutical Biochemistry and Bioanalytics, Pharmaceutical Institute, University of Bonn, Bonn, Germany;3. Molecular, Cellular and Pharmacobiology Section, Institute of Pharmaceutical Biology, University of Bonn, Bonn, Germany;4. Eduard Zintl Institute for Inorganic and Physical Chemistry, Technische Universit?t Darmstadt, Darmstadt, Germany
Abstract:
Keywords:depsipeptides    protein inhibitors    proteins  macrocyclic peptides  NMR spectroscopy
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