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Discovery Process and Characterization of Novel Carbohydrazide Derivatives as Potent and Selective GHSR1a Antagonists
Authors:Fabio Maria Sabbatini Dr.  Romano Di Fabio Dr.  Mauro Corsi Dr.  Paolo Cavanni Dr.  Steve M. Bromidge Dr.  Yves St‐Denis Dr.  Lucilla D'Adamo Dr.  Marilisa Rinaldi Dr.  Chiara Savoia Dr.  Claudia Mundi Dr.  Benedetta Perini Dr.  Andrew J. Carpenter Dr.  Giovanna Dal Forno Dr.  Federico Faggioni Dr.  Michela Tessari Dr.  Francesca Pavone Dr.  Alberto Buson Dr.  Mario Mattioli Dr.  Elisabetta Perdona' Dr.  Sergio Melotto Dr.
Affiliation:1. Neurosciences Center of Excellence for Drug Discovery, GlaxoSmithKline Medicines Research Center, Via A.?Fleming?4, 37135 Verona (Italy), Fax: (+39)?045‐9218196;2. Present address: GlaxoSmithKline, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW (UK);3. Present address: GlaxoSmithKline, 5 Moore Drive, Research Triangle Park, NC 27709 (USA)
Abstract:
Keywords:antagonists  eating disorders  ghrelin  GHSR1a
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