| 邻杂环(噁二唑)甲酰苯胺类化合物的设计合成及杀虫活性初步研究 |
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| 引用本文： | 张湘宁,马海军,张雁南,顾林玲,刘丽,张红芬,俞晓妹,李钰浩,陈凯,倪珏萍.邻杂环(噁二唑)甲酰苯胺类化合物的设计合成及杀虫活性初步研究[J].现代农药,2011,10(3):17-19,23. |
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| 作者姓名： | 张湘宁 马海军 张雁南 顾林玲 刘丽 张红芬 俞晓妹 李钰浩 陈凯 倪珏萍 |
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| 作者单位： | 1. 江苏省农药研究所股份有限公司,南京,210046
2. 南京工业大学理学院,南京,210009 |
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| 基金项目： | 国家"十一五"科技支撑计划 |
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| 摘 要： | 以超高效杀虫剂氯虫苯甲酰胺为先导,在酰胺部分引入了邻杂环(噁二唑),设计并合成了16个含邻杂环(噁二唑)甲酰苯胺类新化合物。生测结果表明,化合物普遍具有高杀虫活性,在10 mg/L剂量下对小菜蛾的致死率均大于80%。本研究结果为该类化合物的创制提供了参考。
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| 关 键 词： | 邻杂环(噁二唑)甲酰苯胺类 合成 杀虫活性 |
Design & Synthesis and Insecticidal Activity of Oxadiazole Benzamide Derivatives |
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| ZHANG Xiang-ning,MA Hai-jun,ZHANG Yan-nan,GU Lin-ling,LIU Li,ZHANG Hong-fen,YU Xiao-mei,LI Yu-hao,CHENG Kai,Ni Jue-ping.Design & Synthesis and Insecticidal Activity of Oxadiazole Benzamide Derivatives[J].Modern Agrochemicals,2011,10(3):17-19,23. |
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| Authors: | ZHANG Xiang-ning MA Hai-jun ZHANG Yan-nan GU Lin-ling LIU Li ZHANG Hong-fen YU Xiao-mei LI Yu-hao CHENG Kai Ni Jue-ping |
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| Affiliation: | ZHANG Xiang-ning1,MA Hai-jun1,ZHANG Yan-nan1,GU Lin-ling1,LIU Li1,ZHANG Hong-fen1,YU Xiao-mei1,LI Yu-hao2,CHENG Kai2,Ni Jue-ping1(1.Jiangsu Pesticide Research Institute Co.,Ltd.,Nanjing 210047,China,2.College of Sciences,Nanjing University of Technology,Nanjing 210009,China) |
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| Abstract: | Excellent insecticide,chlorantranilipeole,was used by leading compound and sixteen novel 3-bromo-N-4-X-2-methyl-6-oxadiazole]-1-(3-chloro-2-pyridinyl)-1H-pyrazole-5-carboxamide derivatives were designed and synthesi-zed.The preliminary bioassay showed that all compounds exhibited good insecticidal activity against Diamondback moth.The death rates were above 80 percent after 3day by feeding containing-pesticide leaf at 10mg/L.It was useful for research of oxadiazole benzamide derivatives. |
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| Keywords: | oxadiazole benzamide derivatives design synthesize insecticidal activity |
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