| 7-取代吲哚类化合物合成及官能团化研究进展 |
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| 引用本文： | 毕维笳,李小军,张国亮,张凤宝.7-取代吲哚类化合物合成及官能团化研究进展[J].化学工业与工程,2007,24(5):446-452. |
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| 作者姓名： | 毕维笳 李小军 张国亮 张凤宝 |
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| 作者单位： | 天津大学化工学院,天津,300072 |
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| 摘 要： | 7-取代吲哚化合物是合成药物及精细化学品的重要中间体.本文综述了近15年金属Pd催化的7-取代吲哚化合物的制备方法,将其分成直接合成法和吲哚7位官能团化法两类,对每一类的反应过程和机理进行了详细介绍和评述.
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| 关 键 词： | Pd 催化 7-取代吲哚 制备 官能团化 吲哚类化合物 直接合成法 官能团化 研究进展 Palladium Indole Functionalization Synthesis 机理 反应过程 方法 催化 金属 重要中间体 精细化学品 药物 取代吲哚化合物 |
| 文章编号： | 1004-9533（2007）05-0446-07 |
| 收稿时间： | 2006-05-29 |
| 修稿时间： | 2006年5月29日 |
Progress in Synthesis and Functionalization of 7-Substituted Indole Catalyzed by Palladium |
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| BI Wei-jia,LI Xiao-jun,ZHANG Guo-liang,ZHANG Feng-bao.Progress in Synthesis and Functionalization of 7-Substituted Indole Catalyzed by Palladium[J].Chemical Industry and Engineering,2007,24(5):446-452. |
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| Authors: | BI Wei-jia LI Xiao-jun ZHANG Guo-liang ZHANG Feng-bao |
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| Affiliation: | School of Chemical Engineering and Technology, Tianjin University, Tianjin 300072, China |
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| Abstract: | 7-substituted indole is key intermediates for forming synthetic drugs and fine chemicals.In this paper,the progresses in preparation methods of 7-substituted indole through palladium-catalyzed reactions in recent 15 years were reviewed.These methods are divided into two categories: the direct synthesis from substituted benzenoid derivatives and the functionalization of performed indoles ring,both of which are introduced in detail in the aspects of mechanism and the processes of reactions. |
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| Keywords: | palladium catalyses 7-substituted indole preparation functionalization |
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