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Tandem Gold(III)‐Catalyzed Amination‐Intramolecular Hydroamination Reactions of 1‐En‐4‐yn‐3‐ols with Sulfonamides: Efficient Approach to Highly Substituted Pyrroles |
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| Authors: | Xing‐Zhong Shu Xue‐Yuan Liu Hui‐Quan Xiao Ke‐Gong Ji Li‐Na Guo Yong‐Min Liang |
| Abstract: | A simple, convenient and efficient synthetic approach to highly substituted pyrroles has been developed by utilizing a gold(III)‐catalyzed tandem amination‐intramolecular hydroamination reaction. The first examples of gold‐catalyzed, selective amination of 1‐en‐4‐yn‐3‐ols have also been disclosed. |
| Keywords: | amination 1‐en‐4‐yn‐3‐ols gold hydroamination pyrroles |