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Computer‐Aided Design,Synthesis and Validation of 2‐Phenylquinazolinone Fragments as CDK9 Inhibitors with Anti‐HIV‐1 Tat‐Mediated Transcription Activity
Authors:Dr. Luca Sancineto  Dr. Nunzio Iraci  Dr. Serena Massari  Dr. Vanessa Attanasio  Dr. Gianmarco Corazza  Dr. Maria Letizia Barreca  Dr. Stefano Sabatini  Dr. Giuseppe Manfroni  Dr. Nilla Roberta Avanzi  Prof. Violetta Cecchetti  Prof. Christophe Pannecouque  Prof. Alessandro Marcello  Dr. Oriana Tabarrini
Affiliation:1. Department of Chemistry and Technology of Drugs, University of Perugia, 06123 Perugia (Italy);2. Molecular Virology Group, International Centre for Genetic Engineering and Biotechnology (ICGEB), 34012 Trieste (Italy);3. Nerviano Medical Sciences, 20014 Nerviano (Italy);4. Rega Institute for Medical Research, Katholieke Universiteit Leuven, 3000 Leuven (Belgium)
Abstract:
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