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Inside Cover: Pentacycloundecane‐diol‐Based HIV‐1 Protease Inhibitors: Biological Screening, 2D NMR,and Molecular Simulation Studies (ChemMedChem 6/2012)
Authors:Dr. Bahareh Honarparvar  Dr. Maya M. Makatini  Sachin A. Pawar  Dr. Katja Petzold  Dr. Mahmoud E. S. Soliman  Prof. Per I. Arvidsson  Dr. Yasien Sayed  Dr. Thavendran Govender  Dr. Glenn E. M. Maguire  Prof. Hendrik G. Kruger
Affiliation:1. School of Chemistry, University of KwaZulu‐Natal, Durban 4001 (South Africa);2. School of Pharmacy and Pharmacology, University of KwaZulu‐Natal, Durban 4001 (South Africa);3. Department of Pharmaceutical Organic Chemistry, Zagazig University, Zagazig 44519 (Egypt);4. Organic Pharmaceutical Chemistry, Uppsala Biomedical Centre, Uppsala University, Box 574, 751?23 Uppsala (Sweden);5. Project Management, CNSP iMed, AstraZeneca R?&?D S?dert?lje, V?stra M?larehamnen 9, 151?85 S?dert?lje (Sweden);6. Protein Structure–Function Research Unit, School of Molecular and Cell Biology, University of the Witwatersrand, Wits 2050 (South Africa)
Abstract:
Keywords:HIV‐1 protease  inhibitors  molecular docking  peptides  transition‐state analogues
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